Benztropine mesylate (苯托品甲磺酸盐) is a dopamine transporter (DAT) inhibitor with IC50 of 118 nM.

Trazodone hydrochlorideis an antidepressant belonging to the class of serotonin receptor antagonists and reuptake inhibitors for treatment of anxiety disorders.

Citalopram HBr, an antidepressant, is an orally administered selective serotonin reuptake inhibitor (SSRI) with IC50 of 1.8 nM.

Zolmitriptan is a novel and highly selective 5-HT(1B/1D) receptor agonist, used in the treatment of acute migraines.

Formoterol Fumarate Dihydrate is a potent, selective and long-acting β2-adrenoceptor agonist used in the management of asthma and chronic obstructive pulmonary disease(COPD).

Agomelatine is classified as a norepinephrine-dopamine disinhibitor (NDDI) due to its antagonism of the 5-HT2C receptor.

Acrivastine is a short-acting histamine 1 receptor antagonist.

Desloratadine is a potent antagonist for  human histamine H1 receptor with IC50 of 51 nM.