Bafilomycin A1 is a vacuolar H+-ATPase inhibitor.

Ataluren selectively induces ribosomal read-through of premature but not normal termination codons.

Ivacaftor is a selective potentiator of CFTR targeting G551D-CFTR and F508del-CFTR.

Lumacaftor acts to correct CFTR mutations common in cystic fibrosis by increasing mutant CFTR (F508del-CFTR) maturation.

Selinexor is an orally bioavailable selective CRM1 inhibitor.

KPT-185 is a selective CRM1 inhibitor.

Andarine is a selective non-steroidal androgen receptor (AR) agonist with Ki of 4 nM, tissue-selective for anabolic organs.

MK-2866 (GTx-024) is a selective androgen receptor modulator (SARM) with Ki of 3.8 nM, and is tissue-selective for anabolic organs.