SRPIN340 is a selective SRPK inhibitor with Ki of 0.89 μM for SRPK1, showing no significant inhibitory activity against more than 140 other kinases..
4μ8C is a potent and selective IRE1 Rnase inhibitor with IC50 of 76 nM.
SF1670 is a highly potent and specific PTEN inhibitor with IC50 of 2 μM.
AZD3965 is a potent, selective and orally available monocarboxylate transporter 1 (MCT1) inhibitor with a binding affinity of 1.6 nM, 6-fold selective over MCT2.
BRD7552 is an inducer of transcription factor PDX1, which increases insulin .
4EGI-1 is a competitive eIF4E/eIF4G interaction inhibitor by binding to eIF4E with KD of 25 μM.
4E1RCat is a dual inhibitor of eIF4E:eIF4G and eIF4E:4E-BP1 interaction, and inhibits the binding of eIF4G to eIF4E with IC50 of 3.2 μM.
Phosphoramidon Disodium Salt is a metalloendopeptidase inhibitor, widely used as a biochemical tool.