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TG003
TS3004-5MG
In-stock
120
- +
TS3004-10MG
200
TS3004-25MG
340
l General Information
Product Name
General description
TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor with IC50 of 20 nM, 200 nM, and 15 nM for Clk1, Clk2, and Clk4, respectively. No inhibitory effect on Clk3, SRPK1, SRPK2, or PKC.
Synonym
(1Z)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one
Purity
≥98.5%(HPLC)
CAS Number
300801-52-9
Formula
C13H15NO2S
Molecular Weight
249.33
Suitability
BioReagent, suitable for cell culture, etc.
l Physical and Chemical Information
Appearance
White to beige Solid
Solubility(25°C)
DMSO
≥45mg/ml
Ethanol
Water
Very slightly soluble
l Storage
Storage temp.
-20°C
l Precautions and Disclaimer
This product is for R&D use only, not for drug, household, or other uses.
l References
1. http://www.drugbank.ca
2. https://ncit.nci.nih.gov
3. https://www.ncbi.nlm.nih.gov