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AZD1080
TS2929-2MG
In-stock
160
- +
TS2929-5MG
200
TS2929-10MG
360
l General Information
Product Name
General description
AZD1080 is a selective, orally active, brain permeable GSK3 inhibitor, inhibits human GSK3α and GSK3β with Ki of 6.9 nM and 31 nM, respectively, shows >14-fold selectivity against CDK2, CDK5, CDK1 and Erk2.
Synonym
AK198951; KB-160506; 2-hydroxy-3-[5-(morpholin-4-ylmethyl)pyridin-2-yl]-1~{H}-indole-5-carbonitrile
Purity
≥98.5%(HPLC)
CAS Number
612487-72-6
Formula
C19H18N4O2
Molecular Weight
334.37
Suitability
BioReagent, suitable for cell culture, etc.
l Physical and Chemical Information
Appearance
Solid
Solubility(25°C)
DMSO
≥45mg/ml
Ethanol
Insoluble
Water
Very slightly soluble
l Storage
Storage temp.
-20°C
l Precautions and Disclaimer
This product is for R&D use only, not for drug, household, or other uses.
l References
1. http://www.drugbank.ca
2. https://ncit.nci.nih.gov
3. https://www.ncbi.nlm.nih.gov
