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CP-724714
TS0519-5MG
In-stock
180
- +
TS0519-10MG
340
l General Information
Product Name
General description
CP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM, >640-fold selectivity against EGFR, InsR, IRG-1R, PDGFR, VEGFR2, Abl, Src, c-Met etc in cell-free assays.
Synonym
ethyl N-[(E)-3-[4-[3-methyl-4-(6-methylpyridin-3-yl)oxyanilino]quinazolin-6-yl]prop-2-enyl]carbamate
Purity
≥98.0%(HPLC)
CAS Number
537705-08-1
Formula
C27H27N5O3
Molecular Weight
469.545
Suitability
BioReagent, suitable for cell culture, etc.
l Physical and Chemical Information
Appearance
Solid
Solubility(25°C)
DMSO
≥50mg/ml
Ethanol
Water
Very slightly soluble
l Storage
Storage temp.
-20°C
l Precautions and Disclaimer
This product is for R&D use only, not for drug, household, or other uses.
l References
1. http://www.drugbank.ca
2. https://ncit.nci.nih.gov
3. https://www.ncbi.nlm.nih.gov
