l General Information |
Product Name | ORY-1001 (RG-6016) 2HCl |
General description | ORY-1001 2HCl is an orally active and selective lysine-specific demethylase LSD1/KDM1A inhibitor. |
Synonym | 4-N-[(1R,2S)-2-phenylcyclopropyl]cyclohexane-1,4-diamine; dihydrochloride |
Purity | ≥98.0%(HPLC) | CAS Number | 1431326-61-2 |
Formula | C15H24Cl2N2 | Molecular Weight | 303.27 |
Suitability | BioReagent, suitable for cell culture, etc. |
l Physical and Chemical Information |
Appearance | solid |
Solubility(25℃) | DMSO | ~5mg/mL |
Ethanol | ~4mg/mL(warmed) |
Water | ≥50mg/mL |
l Biological Information |
Biochem/Physiol
Actions | ORY-1001 2HCl is an orally active and selective lysine-specific demethylase LSD1/KDM1A inhibitor with IC50 of <20 nM, with high selectivity against related FAD dependent aminoxidases. |
l Storage |
Storage temp. | -20℃ |
l Precautions and Disclaimer |
This product is for R&D use only, not for drug, household, or other uses. |
l References |
1. http://www.drugbank.ca 2. https://ncit.nci.nih.gov 3. https://www.ncbi.nlm.nih.gov |
