Product Name

GSK2256098

General description

GSK2256098 is a potent, selective, reversible, and ATP competitive FAK kinase inhibitor.

Synonym

2-[[5-chloro-2-[(5-methyl-2-propan-2-ylpyrazol-3-yl)amino]pyridin-4-yl]amino]-N-methoxybenzamide; GSK-2256098

Purity

≥98%(HPLC)

CAS Number

1224887-10-8

Formula

C²⁰H²³ClN⁶O²

Molecular Weight

414.894

Suitability

BioReagent, suitable for cell culture, etc.

l  Physical and Chemical Information

Appearance

White to Light Yellow solid

Solubility(25℃)

DMSO

≥50mg/mL

Ethanol

≥50mg/mL

Water

Insoluble

l  Biological Information

Biochem/Physiol   Actions

GSK2256098 is a potent, selective, reversible, and ATP competitive FAK kinase inhibitor with apparent Ki of 0.4 nM.

l  Packaging & Storage

Packaging

5mg; 25mg

Storage temp.

-20℃

l  Precautions and Disclaimer

This   product is for R&D use only, not for drug, household, or other uses.

l  References

1.    http://www.drugbank.ca

2.    https://ncit.nci.nih.gov

3.    https://www.ncbi.nlm.nih.gov